tallózása szerző szerint "SE/GYTK/Szerves Vegytani Intézet"

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(3Z)-3-(2-[4-(aryl)-1,3-thiazol-2-yl]hydrazin-1-ylidene)-2,3-dihydro-1H-indol-2-one derivatives as dual inhibitors of HIV-1 reverse transcriptase.

Meleddu Rita,; Distinto Simona,; Corona Angela,; Bianco Giulia,; Cannas Valeria,; Mátyus, Péter; Bogdán, Dóra (2015)

The HIV-1 Reverse Transcriptase (RT) is a validated and deeply explored biol. target for the treatment of AIDS. However, only drugs targeting the RT-assocd. DNA polymerase (DP) function have been approved for clin. use. ...
Analgesic and Anti-Inflammatory Effects of the Novel Semicarbazide-Sensitive Amine-Oxidase Inhibitor SzV-1287 in Chronic Arthritis Models of the Mouse.

Horváth Ádám; Menghis A; Botz Bálint; Borbély Éva; Kemény Ágnes; Tékus Valéria; Csepregi Janka Zsófia; Mócsai Attila; Juhász Tamás; Zákány Róza; Bogdán Dóra; Mátyus Péter; Keeble J; Pintér Erika; Helyes Zsuzsanna (2017)

Semicarbazide-sensitive amine oxidase (SSAO) catalyses oxidative deamination of primary amines. Since there is no data about its function in pain and arthritis mechanisms, we investigated the effects of our novel SSAO ...
Analgesic effects of the novel semicarbazide-sensitive amine oxidase inhibitor SZV 1287 in mouse pain models with neuropathic mechanisms: involvement of transient receptor potential vanilloid 1 and ankyrin 1 receptors.

Horvath, A; Tekus, V; Bencze, N; Szentes, N; Scheich, B; Bolcskei, K; Szoke, E; Mócsai, Attila; Toth-Sarudy, E; Mátyus, Péter; Pinter, E; Helyes, Z (2018)

Semicarbazide-sensitive amine oxidase (SSAO) produces tissue irritants by deamination of primary amines, which activate transient receptor potential ankyrin 1 (TRPA1) and vanilloid 1 (TRPV1) receptors expressed predominantly ...
Analysis of Edg-Like LPA Receptor-Ligand Interactions

Balogh, Balázs; Pazmany Tamas,; Mátyus, Péter (2015)

The phospholipid derivative lysophosphatidic acid (LPA) serves as a signalling molecule through the activation of LPA receptors, which belong to the G-protein-coupled receptors. From a pharmacological point of view, the ...
Anti-inflammatory effects of a triple-bond resveratrol analog: Structure and function relationship

Antus, Csenge Petra; Radnai, Balázs; Dombovari Peter,; Fónai, Fruzsina; Avar, Péter Ágoston; Mátyus, Péter; Rácz, Boglárka; Sümegi, Balázs; Veres, Balázs (2015)
Chemically Modified Derivatives of the Activator Compound Cloxyquin Exert Inhibitory Effect on TRESK (K2P18.1) Background Potassium Channel.

Lengyel, Miklós; Erdélyi, Ferenc; Pergel, Enikő; Bálint-Polonka, Ágnes; Dobolyi, Alice; Bozsaki, Péter; Dux, Mária; Király, Kornél; Hegedűs, Tamás; Czirják, Gábor; Mátyus, Péter; Enyedi, Péter (2019)

Cloxyquin has been reported as a specific activator of TRESK (K2P18.1, TWIK-related spinal cord K+ channel) background potassium channel. In this study, we have synthetized chemically modified analogues of cloxyquin and ...
CYP24A1 inhibition facilitates the anti-tumor effect of vitamin D3 on colorectal cancer cells

Kósa János; Horváth P; Wölfling János; Kovács Dóra Irén; Balla Bernadett; Mátyus Péter; Horváth Evelin; Speer Gábor; Takács István; Nagy Zsolt; Horváth Henrik Csaba; Lakatos Péter (2013)

AIM: The effects of vitamin D3 have been investigated on various tumors, including colorectal cancer (CRC). 25-hydroxyvitamin-D3-24-hydroxylase (CYP24A1), the enzyme that inactivates the active vitamin D3 metabolite ...
Determination of circular dichroism and ultraviolet spectral parameters of norgestimate- and other Δ4-3-ketosteroid Oxime isomers via normal phase HPLC method

Szentesi A; Gergely András; Horváth Péter; Mahó S; Mátyus Péter; Szász György (2001)
Encoding Information into Polyethylene Glycol Using an Alcohol-Isocyanate “Click” Reaction

Nagy, Lajos; Kuki, Ákos; Nagy, Tibor; Vadkerti, Bence; Erdélyi, Zoltán; Kárpáti, Levente; Zsuga, Miklós; Kéki, Sándor (2020)

In this article, the capability of encoding information using a homologous series of monodisperse monomethoxypolyethylene glycols (mPEG), with a number of ethylene oxide units ranging from nEO = 5 to 8, and monodisperse ...
Equilibrium, structural and antibacterial characterization of moxifloxacin-β-cyclodextrin complex

Szabó Zoltán-István; Deme Ruth; Mucsi Zoltán; Rusu Aura; Mare Anca Delia; Tóth Gergő (2018)

Moxifloxacin (MOX), a novel fourth-generation fluoroquinolone antibacterial was characterized in terms of β-cyclodextrin (β-CD) complexation in order to improve its antibacterial activity. The inclusion complexation has ...
Flow-chemistry enabled efficient synthesis of β-peptides: backbone topology vs. helix formation

Nekkaa, Imane; Bogdán, Dóra; Gáti, Tamás; Béni, Szabolcs; Juhász, Tünde; Palkó, Márta; Paragi, Gábor; Tóth, Gábor K.; Fülöp, Ferenc; Mándity, István M. (2019)

Enantiodiscriminative helix formation was observed for beta-peptide H14 helices. This observation is caused by the synperiplanar orientation of H-O atoms which is more unfavorable than those for H-H interaction. The 1,2 ...
Functionalization of the pyridazin-3(2H)-one ring via palladium-catalysed aminocarbonylation

Takács Attila; Czompa Andrea; Krajsovszky Gábor; Mátyus Péter; Kollár László (2012)
Galls of European Fraxinus trees as new and abundant sources of valuable phenylethanoid and coumarin glycosides

Zürn, M.; Tóth, Gergő; Mazákné Kraszni, Márta; Sólyomváry, Anna; Mucsi, Zoltán; Deme, Ruth; Rózsa, B.; Fodor, Blanka; Molnár-Perl, Ibolya; Horváti, Kata; Bősze, Szilvia; Pályi, B.; Kis, Z.; Béni, Szabolcs; Noszál, Béla; Boldizsár, Ime (2019)
Imidazoline versus alpha2-adrenoceptors in the control of gastric motility in mice

Zádori Zoltán Sándor; Fehér Ágnes; Al-Khrasani Mahmoud; Lackó Erzsébet; Tóth Viktória; Mátyus Péter; Gyires Klára (2013)
'Interrupted' diazotization of 3-aminoindoles and 3-aminopyrroles

Parrino Barbara,; Spano Virginia,; Carbone Anna,; Montalbano Alessandra,; Barraja Paola,; Mátyus, Péter (2014)
Lack of association between VAP-1/SSAO activity and corneal neovascularization in a rabbit model

Énzsöly Anna; Markó Katalin; Tábi Tamás; Szökő Éva; Zelkó Romána; Tóth Miklós; Mátyus Péter; Németh János Tibor (2013)
Mechanisms of glycine release, which build up synaptic and extrasynaptic glycine levels

Hársing, László Gábor; Mátyus, Péter (2013)

84875595371
Multi-aspect candidates for repositioning: data fusion methods using heterogeneous information sources.

Arany Ádám; Bolgar B; Balogh Balázs; Antal P; Mátyus Péter (2013)

Drug repositioning, an innovative therapeutic application of an old drug, has received much attention as a particularly costeffective strategy in drug R&D Recent work has indicated that repositioning can be promoted by ...
New computational studies to support cyclin-dependent kinase 9 inhibitor screening and design

Fábián, Márk; Balogh, Balázs; Czudor, Zsófia; Örfi, László (2019)
Novel 1,4-benzoxazine and 1,4-benzodioxine inhibitors of angiogenesis.

Ilić M; Ilaš J; Dunkel Petra; Mátyus Péter; Bohác A (2012)

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